Assay Report Card

Basic Information

ID: ALA3578424

Type: Functional

Description: Ex vivo histamine H3 receptor occupancy in Sprague-Dawley rat striatum at 3 mg/kg, po measured at 1 hr by autoradiographic analysis

Organism: Rattus norvegicus

Strain: Sprague-Dawley

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
329.492.842.84
447.531.681.68
343.471.831.83
365.911.441.44
347.482.792.79
345.462.542.54