Assay Report Card

Basic Information

ID: ALA3579924

Type: Binding

Description: Orthosteric non-competitive inhibition of human ASIC1a endogenously expressed in HEK293 cells clamped at -100 mV gated ionic current assessed as maximal evoked response for steady-state activation at 100 nM by standard whole cell patch clamp assay relative to untreated control

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
426.954.084.08