Basic Information
ID: ALA3591169
Type: Functional
Description: Antagonist activity against CB1R (unknown origin) CHO cells stably expressing Galpha16 assessed as inhibition of CP55940-induced increase in intracellular calcium level pre-treated 10 mins before CP55940 stimulation by microplate reader based assay
Format: BAO_0000219
Organism: Homo sapiens
Cell type: CHO
Target: Cannabinoid CB1 receptor(ALA218)
Document: ALA3588836
Antagonist activity against CB1R (unknown origin) CHO cells stably expressing Galpha16 assessed as inhibition of CP55940-induced increase in intracellular calcium level pre-treated 10 mins before CP55940 stimulation by microplate reader based assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA3591169
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 463.80 | 5.94 | 5.94 |
| 409.49 | 3.27 | 3.27 |
| 354.49 | 4.52 | 4.52 |
| 370.49 | 4.22 | 4.22 |
| 374.91 | 4.87 | 4.87 |
| 384.52 | 4.53 | 4.53 |
| 388.94 | 5.17 | 5.17 |
| 400.52 | 4.23 | 4.23 |
| 422.57 | 4.86 | 4.86 |
| 426.99 | 5.50 | 5.50 |
| 436.60 | 5.17 | 5.17 |
| 356.47 | 3.83 | 3.83 |
| 370.49 | 4.22 | 4.22 |
| 384.52 | 4.61 | 4.61 |
| 354.49 | 4.52 | 4.52 |
| 396.58 | 5.51 | 5.51 |
| 424.46 | 5.11 | 5.11 |
| 374.91 | 4.87 | 4.87 |
| 419.36 | 4.97 | 4.97 |
| 408.46 | 5.23 | 5.23 |