Basic Information
ID: ALA3591195
Type: Functional
Description: Immediate antagonist/Inverse agonist activity at hemagglutinin-tagged human CB1 receptor expressed in HEK293 cells assessed as reversal of 1 uM CP55,940-induced inhibition of 5 uM forskolin-induced cAMP accumulation by kinetic cAMP assay
Format: BAO_0000219
Organism: Homo sapiens
Cell type: HEK293
Target: Cannabinoid CB1 receptor(ALA218)
Document: ALA3588815
Immediate antagonist/Inverse agonist activity at hemagglutinin-tagged human CB1 receptor expressed in HEK293 cells assessed as reversal of 1 uM CP55,940-induced inhibition of 5 uM forskolin-induced cAMP accumulation by kinetic cAMP assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA3591195
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 463.80 | 5.94 | 5.94 |
| 340.85 | 4.66 | 4.66 |
| 361.27 | 5.01 | 5.01 |
| 344.82 | 4.50 | 4.50 |
| 375.52 | 4.69 | 4.69 |
| 343.77 | 3.70 | 3.70 |
| 356.85 | 4.82 | 4.82 |