Basic Information
ID: ALA3607765
Type: Binding
Description: Inhibition of human recombinant Histidine-tagged RSK2 using biotin-AGAGRSRHSSYPAGT-OH as substrate preincubated for 30 mins followed by ATP and substrate addition measured after 180 mins by AlphaScreen assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA3607765
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 252.27 | 3.15 | 3.15 |
| 236.27 | 3.45 | 3.45 |
| 236.27 | 3.45 | 3.45 |
| 251.29 | 3.03 | 3.03 |
| 288.25 | 3.43 | 3.43 |
| 263.30 | 3.83 | 3.83 |
| 299.28 | 4.11 | 4.11 |
| 283.28 | 4.40 | 4.40 |
| 291.30 | 3.63 | 3.63 |
| 290.31 | 3.20 | 3.20 |
| 249.26 | 3.86 | 3.86 |
| 297.30 | 4.71 | 4.71 |
| 313.30 | 4.41 | 4.41 |
| 342.35 | 3.74 | 3.74 |
| 349.34 | 4.79 | 4.79 |
| 368.38 | 4.24 | 4.24 |
| 381.43 | 4.15 | 4.15 |
| 301.27 | 4.54 | 4.54 |
| 297.30 | 4.71 | 4.71 |
| 313.30 | 4.41 | 4.41 |
| 340.33 | 3.76 | 3.76 |
| 367.40 | 3.81 | 3.81 |
| 381.43 | 4.15 | 4.15 |
| 368.38 | 4.24 | 4.24 |
| 314.29 | 3.80 | 3.80 |
| 334.18 | 5.57 | 5.57 |
| 396.44 | 3.73 | 3.73 |
| 410.47 | 4.19 | 4.19 |
| 452.55 | 5.22 | 5.22 |
| 486.57 | 6.20 | 6.20 |
| 313.31 | 3.69 | 3.69 |
| 327.33 | 4.14 | 4.14 |
| 355.39 | 4.92 | 4.92 |
| 439.51 | 4.37 | 4.37 |
| 391.42 | 3.42 | 3.42 |