Basic Information
ID: ALA3610932
Type: Binding
Description: Inhibition of wild type dephosphorylated form of PAK1 (249 to 545) (unknown origin) expressed in Escherichia coli using 5-Fluo-Ahx-AKRRRLSSLRA-COOH as substrate preincubated for 60 mins followed by substrate addition measured after 60 mins by Caliper assay
Format: BAO_0000019
Organism: Homo sapiens
Target: Serine/threonine-protein kinase PAK 1(ALA4600)
Document: ALA3608218
Inhibition of wild type dephosphorylated form of PAK1 (249 to 545) (unknown origin) expressed in Escherichia coli using 5-Fluo-Ahx-AKRRRLSSLRA-COOH as substrate preincubated for 60 mins followed by substrate addition measured after 60 mins by Caliper assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA3610932
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 328.37 | 3.35 | 3.35 |
| 358.85 | 3.89 | 3.89 |
| 372.88 | 4.28 | 4.28 |
| 458.97 | 5.63 | 5.63 |
| 457.98 | 5.20 | 5.20 |
| 479.93 | 5.06 | 5.06 |