Inhibition of human NET expressed in HEK293 cells assessed as reduction of serotonin reuptake using [3H]-NET at 1 uM after 15 mins by liquid scintilla...

Basic Information

ID: ALA3614495

Type: Binding

Description: Inhibition of human NET expressed in HEK293 cells assessed as reduction of serotonin reuptake using [3H]-NET at 1 uM after 15 mins by liquid scintillation counting relative to GBR-12909

Format: BAO_0000219

Organism: Homo sapiens

Cell type: HEK293

Target:  Norepinephrine transporter(ALA222)

Document:  ALA3611988

Inhibition of human NET expressed in HEK293 cells assessed as reduction of serotonin reuptake using [3H]-NET at 1 uM after 15 mins by liquid scintillation counting relative to GBR-12909: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
405.375.075.07
386.544.914.91
386.544.914.91
465.445.685.68
416.574.924.92
391.344.684.68
373.503.923.92
372.514.524.52
372.514.524.52
451.415.295.29