Inhibition of human NET expressed in HEK293 cells assessed as reduction of serotonin reuptake using [3H]-NET at 3 uM after 15 mins by liquid scintilla...

Basic Information

ID: ALA3614496

Type: Binding

Description: Inhibition of human NET expressed in HEK293 cells assessed as reduction of serotonin reuptake using [3H]-NET at 3 uM after 15 mins by liquid scintillation counting relative to venlafaxine HCl

Format: BAO_0000219

Organism: Homo sapiens

Cell type: HEK293

Target:  Norepinephrine transporter(ALA222)

Document:  ALA3611988

Inhibition of human NET expressed in HEK293 cells assessed as reduction of serotonin reuptake using [3H]-NET at 3 uM after 15 mins by liquid scintillation counting relative to venlafaxine HCl: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
426.605.285.28
375.524.244.24
376.504.514.51
392.574.984.98
412.585.435.43
495.496.596.59
387.534.314.31
361.493.853.85
362.474.124.12
378.544.594.59
398.555.045.04
412.584.894.89
481.476.206.20
402.544.534.53