Basic Information
ID: ALA3619088
Type: Functional
Description: Antagonist activity at human glucagon receptor expressed in HEK293 cell membranes assessed as inhibition of glucagon-stimulated intracellular cAMP formation preincubated for 30 mins followed by glucagon stimulation measured after 5 mins by TR-FRET analysis
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA3619088
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 635.99 | 8.23 | 8.23 |
| 553.87 | 7.80 | 7.80 |
| 602.44 | 7.87 | 7.87 |