Basic Information
ID: ALA3619501
Type: Binding
Description: Inverse agonist activity at GAL4-fused human RORa expressed in HEK293 cells assessed as suppression of basal transcriptional activity after 20 hrs by dual-glo luciferase reporter gene assay
Format: BAO_0000219
Organism: Homo sapiens
Cell type: HEK293
Target: Nuclear receptor ROR-alpha(ALA5868)
Document: ALA3616373
Inverse agonist activity at GAL4-fused human RORa expressed in HEK293 cells assessed as suppression of basal transcriptional activity after 20 hrs by dual-glo luciferase reporter gene assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA3619501
EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 462.90 | 5.01 | 5.01 |
| 446.45 | 4.50 | 4.50 |
| 432.42 | 4.11 | 4.11 |
| 444.92 | 4.87 | 4.87 |