Basic Information
ID: ALA3619994
Type: Binding
Description: Inhibition of recombinant human activated-MMP1 using Mca-Lys-Pro-Leu-Gly-Leu-Dap(Dnp)-Ala-Arg-NH2 as fluorogenic substrate incubated for 4 hrs followed by substrate addition measured every 10 secs for 20 mins by fluorometric assay
Format: BAO_0000357
Organism: Homo sapiens
Target: Matrix metalloproteinase-1(ALA332)
Document: ALA3616369
Inhibition of recombinant human activated-MMP1 using Mca-Lys-Pro-Leu-Gly-Leu-Dap(Dnp)-Ala-Arg-NH2 as fluorogenic substrate incubated for 4 hrs followed by substrate addition measured every 10 secs for 20 mins by fluorometric assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA3619994
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 511.60 | 3.38 | 3.38 |
| 485.58 | 1.50 | 1.50 |
| 449.53 | 2.08 | 2.08 |
| 525.63 | 3.31 | 3.31 |
| 479.56 | 2.09 | 2.09 |
| 555.65 | 3.32 | 3.32 |
| 373.43 | 0.42 | 0.42 |
| 567.62 | 3.25 | 3.25 |