Assay Report Card

Basic Information

ID: ALA3624841

Type: Functional

Description: Antitumor activity against bicalutamide-resistant human CWR22 cells in Balb/c athymic (nu/nu) mouse CWR22-BMSLD1 prostate cancer xenograft model assessed as tumor growth inhibition at 90 mg/kg, po qd administered for 45 days measured from day 10 to 45 during compound dosing

Organism: Homo sapiens

Cell type: CWR22

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
471.461.941.94