Basic Information
ID: ALA3626472
Type: Functional
Description: Antagonist activity at human PKR1 expressed in rat RBL2H3 cells assessed as inhibition of PK1-stimulated intracellular calcium release incubated for 10 mins prior to PK1 stimulation by FLIPR assay
Format: BAO_0000219
Organism: Homo sapiens
Cell type: RBL-2H3
Target: Prokineticin receptor 1(ALA5649)
Document: ALA3621181
Antagonist activity at human PKR1 expressed in rat RBL2H3 cells assessed as inhibition of PK1-stimulated intracellular calcium release incubated for 10 mins prior to PK1 stimulation by FLIPR assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA3626472
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 391.52 | 4.10 | 4.10 |
| 364.49 | 4.46 | 4.46 |
| 349.44 | 3.33 | 3.33 |
| 385.90 | 3.65 | 3.65 |
| 362.84 | 3.58 | 3.58 |
| 363.85 | 2.14 | 2.14 |