Basic Information
ID: ALA3626890
Type: Binding
Description: Inhibition of recombinant human KAT2A using biotinylated histone H3 (1 to 21 amino acid residues) as substrate at 50 uM preincubated for 10 mins followed by acetyl-CoA addition measured after 10 mins by time resolved fluorescence assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA3626890
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 262.72 | 3.10 | 3.10 |
| 246.27 | 2.59 | 2.59 |
| 243.29 | 2.15 | 2.15 |
| 347.83 | 3.37 | 3.37 |
| 234.31 | 2.51 | 2.51 |
| 360.46 | 2.84 | 2.84 |
| 292.36 | 3.91 | 3.91 |
| 299.35 | 3.23 | 3.23 |
| 284.37 | 3.66 | 3.66 |
| 248.33 | 2.82 | 2.82 |
| 365.37 | 4.15 | 4.15 |
| 360.48 | 5.46 | 5.46 |
| 276.75 | 3.16 | 3.16 |
| 311.19 | 3.81 | 3.81 |
| 310.30 | 3.53 | 3.53 |
| 385.45 | 3.96 | 3.96 |
| 291.36 | 2.16 | 2.16 |
| 290.37 | 2.82 | 2.82 |
| 295.36 | 1.82 | 1.82 |
| 313.43 | 3.16 | 3.16 |
| 266.32 | 1.64 | 1.64 |
| 237.28 | 1.93 | 1.93 |
| 285.32 | 2.74 | 2.74 |
| 278.38 | 2.23 | 2.23 |
| 264.35 | 1.84 | 1.84 |
| 266.32 | 0.83 | 0.83 |
| 299.36 | 1.77 | 1.77 |
| 324.43 | 4.48 | 4.48 |