Basic Information
ID: ALA3626893
Type: Binding
Description: Inhibition of recombinant human CBP using biotinylated histone H3 (1 to 21 amino acid residues) as substrate preincubated for 10 mins followed by acetyl-CoA addition measured after 10 mins by time resolved fluorescence assay
Format: BAO_0000357
Organism: Homo sapiens
Target: CREB-binding protein(ALA5747)
Document: ALA3621044
Inhibition of recombinant human CBP using biotinylated histone H3 (1 to 21 amino acid residues) as substrate preincubated for 10 mins followed by acetyl-CoA addition measured after 10 mins by time resolved fluorescence assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA3626893
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 262.72 | 3.10 | 3.10 |
| 246.27 | 2.59 | 2.59 |
| 347.83 | 3.37 | 3.37 |
| 276.75 | 3.16 | 3.16 |
| 311.19 | 3.81 | 3.81 |
| 310.30 | 3.53 | 3.53 |
| 385.45 | 3.96 | 3.96 |
| 295.36 | 1.82 | 1.82 |
| 313.43 | 3.16 | 3.16 |