ID: ALA3626894
Type: Binding
Description: Inhibition of recombinant human p300 using biotinylated histone H3 (1 to 21 amino acid residues) as substrate at 50 uM preincubated for 10 mins followed by acetyl-CoA addition measured after 10 mins by time resolved fluorescence assay
Organism: Homo sapiens
Bioactivity
Activity Types for Assay ALA3626894
Inhibition
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
262.72 | 3.10 | 3.10 |
246.27 | 2.59 | 2.59 |
243.29 | 2.15 | 2.15 |
347.83 | 3.37 | 3.37 |
234.31 | 2.51 | 2.51 |
360.46 | 2.84 | 2.84 |
292.36 | 3.91 | 3.91 |
299.35 | 3.23 | 3.23 |
284.37 | 3.66 | 3.66 |
248.33 | 2.82 | 2.82 |
365.37 | 4.15 | 4.15 |
360.48 | 5.46 | 5.46 |
276.75 | 3.16 | 3.16 |
311.19 | 3.81 | 3.81 |
310.30 | 3.53 | 3.53 |
385.45 | 3.96 | 3.96 |
291.36 | 2.16 | 2.16 |
290.37 | 2.82 | 2.82 |
295.36 | 1.82 | 1.82 |
313.43 | 3.16 | 3.16 |
266.32 | 1.64 | 1.64 |
237.28 | 1.93 | 1.93 |
285.32 | 2.74 | 2.74 |
278.38 | 2.23 | 2.23 |
264.35 | 1.84 | 1.84 |
266.32 | 0.83 | 0.83 |
299.36 | 1.77 | 1.77 |
324.43 | 4.48 | 4.48 |