Assay Report Card

Basic Information

ID: ALA3630622

Type: Binding

Description: Inhibition of poly-histidine tagged full-length rat ARFGAP1 expressed in Sf9 cells assessed as remaining enzyme activity at 20 uM using purified WT ARF1 pre-loaded with [gamm-32P]-labeled GTP incubated for 5 mins before ARF1-GTP addition followed by 25 mins incubation by scintillation counting method

Organism: Rattus norvegicus

Cell type: Sf9

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
491.605.175.17
567.696.846.84
577.697.507.50
553.676.786.78
535.655.345.34
581.727.407.40
597.726.856.85
583.696.966.96
581.727.157.15
585.686.986.98
602.704.824.82
617.674.724.72
558.654.754.75
572.674.814.81
586.705.125.12
571.646.086.08
577.697.507.50
595.637.377.37
557.656.366.36
587.686.376.37
587.686.376.37
465.564.574.57
520.644.394.39
573.708.598.59
577.647.837.83
583.709.259.25
583.709.259.25
601.639.129.12
563.668.118.11
537.677.487.48
541.616.726.72
547.668.148.14
547.668.148.14
565.608.018.01
527.637.007.00
505.626.016.01
509.575.255.25
515.626.676.67
515.626.676.67
613.676.656.65
619.738.078.07
619.738.078.07