Basic Information
ID: ALA3631243
Type: Binding
Description: Inhibition of recombinant mouse 17beta HSD1 expressed in HEK293 cells using unlabeled- and labelled [2,4,6,7-3H]-E1 as substrate at 1 uM incubated for 10 mins by HPLC analysis
Format: BAO_0000219
Organism: Mus musculus
Cell type: HEK293
Target: Estradiol 17-beta-dehydrogenase 1(ALA1914269)
Document: ALA3627664
Inhibition of recombinant mouse 17beta HSD1 expressed in HEK293 cells using unlabeled- and labelled [2,4,6,7-3H]-E1 as substrate at 1 uM incubated for 10 mins by HPLC analysis: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA3631243
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 312.37 | 5.59 | 5.59 |
| 286.33 | 4.63 | 4.63 |
| 296.35 | 4.06 | 4.06 |
| 314.34 | 4.20 | 4.20 |
| 310.37 | 4.37 | 4.37 |
| 492.56 | 6.26 | 6.26 |
| 289.29 | 3.08 | 3.08 |
| 285.32 | 3.25 | 3.25 |
| 288.30 | 3.68 | 3.68 |
| 295.36 | 3.93 | 3.93 |
| 295.36 | 3.93 | 3.93 |
| 435.53 | 5.15 | 5.15 |
| 598.42 | 6.81 | 6.81 |
| 460.54 | 5.02 | 5.02 |
| 435.53 | 5.15 | 5.15 |
| 598.42 | 6.81 | 6.81 |
| 460.54 | 5.02 | 5.02 |
| 441.56 | 5.21 | 5.21 |
| 451.53 | 4.86 | 4.86 |
| 415.47 | 5.31 | 5.31 |
| 429.50 | 5.33 | 5.33 |
| 460.54 | 5.02 | 5.02 |
| 480.52 | 5.06 | 5.06 |
| 480.52 | 5.06 | 5.06 |
| 480.52 | 5.06 | 5.06 |
| 525.52 | 4.97 | 4.97 |
| 453.52 | 5.29 | 5.29 |
| 453.52 | 5.29 | 5.29 |
| 453.52 | 5.29 | 5.29 |
| 514.42 | 5.92 | 5.92 |
| 550.40 | 6.19 | 6.19 |
| 520.42 | 6.16 | 6.16 |
| 465.55 | 5.16 | 5.16 |
| 492.58 | 5.11 | 5.11 |
| 449.55 | 5.46 | 5.46 |
| 449.55 | 5.46 | 5.46 |
| 483.54 | 5.30 | 5.30 |
| 469.52 | 5.00 | 5.00 |
| 331.34 | 4.21 | 4.21 |
| 634.40 | 7.09 | 7.09 |
| 555.50 | 6.33 | 6.33 |
| 472.49 | 4.83 | 4.83 |
| 475.50 | 4.16 | 4.16 |
| 435.47 | 4.53 | 4.53 |
| 449.55 | 5.46 | 5.46 |
| 364.34 | 5.08 | 5.08 |
| 270.31 | 3.54 | 3.54 |