Inhibition of recombinant rat 17beta HSD1 expressed in HEK293 cells using unlabeled- and labelled [2,4,6,7-3H]-E1 as substrate at 250 nM incubated for...

Basic Information

ID: ALA3631244

Type: Binding

Description: Inhibition of recombinant rat 17beta HSD1 expressed in HEK293 cells using unlabeled- and labelled [2,4,6,7-3H]-E1 as substrate at 250 nM incubated for 10 mins by HPLC analysis

Format: BAO_0000219

Organism: Rattus norvegicus

Cell type: HEK293

Target:  Estradiol 17-beta-dehydrogenase 1(ALA1914267)

Document:  ALA3627664

Inhibition of recombinant rat 17beta HSD1 expressed in HEK293 cells using unlabeled- and labelled [2,4,6,7-3H]-E1 as substrate at 250 nM incubated for 10 mins by HPLC analysis: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
331.344.214.21
634.407.097.09
555.506.336.33
539.506.456.45
472.494.834.83
475.504.164.16
435.474.534.53
449.504.844.84
463.534.874.87