PIM-2 Enzyme Assay: The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of ...

Basic Information

ID: ALA3705115

Type: Binding

Description: PIM-2 Enzyme Assay: The assay for the determination of PIM activity is based on the incorporation of [33P] ATP into PIM2tide substrate and capture of the radiolabeled peptide onto a Whatman P81 (phosphocellulose) filter plate. Assay mixtures contained 4 uM [gamma-33P] ATP (20 uCi/mL), 1.0 uM PIM2tide and 1.5 nM PIM-2 in place of PIM-1.

Format: BAO_0000357

Organism: Homo sapiens

Target:  Serine/threonine-protein kinase PIM2(ALA4523)

Document:  ALA3639321

BindingDB Source:  6019

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
344.423.113.11
400.534.674.67
359.433.663.66
330.402.722.72
330.402.722.72
418.504.274.27
318.382.712.71
388.524.154.15
345.413.083.08
319.372.672.67
331.382.692.69
331.382.692.69
403.442.622.62
359.433.323.32
373.463.863.86
359.433.323.32
359.433.593.59
347.423.313.31
377.452.802.80
347.423.443.44
375.483.913.91
346.393.103.10
332.414.374.37
348.413.343.34
363.403.023.02
363.403.023.02
375.483.963.96
361.453.573.57
371.443.613.61
375.484.094.09
375.484.094.09
361.453.703.70
361.453.703.70
389.504.484.48
389.504.484.48
365.413.453.45
388.432.872.87
355.352.922.92
365.413.453.45
353.393.923.92
353.393.923.92
377.423.413.41
377.423.413.41
359.433.473.47
416.492.532.53
432.482.462.46
375.432.442.44
389.463.093.09
426.324.074.07
381.393.163.16
381.393.163.16
345.413.083.08
336.351.681.68
426.324.074.07
387.494.194.19
423.524.984.98
373.463.713.71
387.494.104.10
413.534.494.49
401.514.354.35
465.564.354.35
375.432.442.44
389.463.093.09
339.364.134.13
354.373.713.71
355.363.113.11
456.324.184.18
442.293.793.79
417.494.294.29
403.463.903.90
453.525.085.08
439.494.694.69
434.482.612.61
391.453.763.76
421.483.123.12
417.513.423.42
381.393.163.16
395.413.553.55
391.453.723.72
399.383.463.46
363.403.023.02
417.494.294.29
391.453.723.72
402.433.963.96
395.413.553.55
395.413.553.55
405.484.154.15
423.474.104.10
395.413.553.55
349.372.632.63
367.362.772.77
407.453.423.42
425.443.563.56
451.503.443.44
396.422.842.84
378.432.702.70
421.483.623.62
465.533.333.33
389.462.832.83
377.423.423.42