Basic Information
ID: ALA3720934
Type: Binding
Description: Inhibition of N-terminal GST-tagged full-length human PBK (1 to 322 residues) using FITC-labeled histone-H3 peptide substrate incubated for 1 hr by fluorescence polarization based assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA3720934
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 411.54 | 1.58 | 1.58 |
| 351.45 | 2.62 | 2.62 |
| 393.52 | 3.47 | 3.47 |
| 299.38 | 1.83 | 1.83 |
| 285.35 | 1.32 | 1.32 |
| 299.38 | 1.56 | 1.56 |
| 341.44 | 2.69 | 2.69 |
| 299.38 | 1.39 | 1.39 |
| 341.44 | 2.42 | 2.42 |
| 313.41 | 2.08 | 2.08 |
| 341.44 | 2.09 | 2.09 |
| 369.49 | 3.18 | 3.18 |
| 411.54 | 1.71 | 1.71 |
| 355.47 | 2.93 | 2.93 |
| 341.44 | 2.42 | 2.42 |
| 327.41 | 2.17 | 2.17 |
| 355.47 | 2.34 | 2.34 |
| 341.44 | 2.42 | 2.42 |
| 412.52 | 1.74 | 1.74 |
| 355.47 | 2.93 | 2.93 |
| 400.51 | 1.60 | 1.60 |
| 327.41 | 2.17 | 2.17 |
| 339.44 | 2.34 | 2.34 |
| 411.54 | 1.58 | 1.58 |
| 404.27 | 2.71 | 2.71 |
| 341.44 | 2.69 | 2.69 |
| 369.49 | 3.18 | 3.18 |
| 397.55 | 3.96 | 3.96 |
| 412.52 | 2.00 | 2.00 |
| 259.31 | 0.69 | 0.69 |
| 313.39 | 1.64 | 1.64 |
| 355.47 | 2.34 | 2.34 |
| 313.39 | 1.78 | 1.78 |
| 413.52 | 3.65 | 3.65 |
| 410.55 | 3.16 | 3.16 |
| 381.52 | 3.36 | 3.36 |
| 355.47 | 2.81 | 2.81 |
| 426.55 | 2.13 | 2.13 |
| 355.42 | 1.73 | 1.73 |
| 341.44 | 2.56 | 2.56 |
| 355.47 | 2.81 | 2.81 |
| 406.31 | 2.93 | 2.93 |
| 338.40 | 2.38 | 2.38 |
| 420.34 | 3.18 | 3.18 |
| 357.44 | 1.58 | 1.58 |
| 311.39 | 1.74 | 1.74 |
| 371.47 | 1.83 | 1.83 |
| 420.34 | 3.18 | 3.18 |
| 369.45 | 1.98 | 1.98 |
| 395.47 | 1.11 | 1.11 |
| 216.29 | 1.49 | 1.49 |
| 355.83 | 2.76 | 2.76 |
| 259.31 | 0.96 | 0.96 |
| 352.42 | 2.77 | 2.77 |
| 412.52 | 1.74 | 1.74 |
| 341.44 | 2.51 | 2.51 |
| 390.24 | 2.46 | 2.46 |
| 327.41 | 2.17 | 2.17 |
| 326.43 | 2.77 | 2.77 |
| 430.53 | 0.96 | 0.96 |
| 245.29 | 0.44 | 0.44 |
| 406.31 | 2.93 | 2.93 |
| 371.47 | 1.83 | 1.83 |
| 369.45 | 1.98 | 1.98 |
| 420.34 | 3.18 | 3.18 |
| 420.34 | 3.32 | 3.32 |
| 298.42 | 3.22 | 3.22 |
| 340.45 | 3.02 | 3.02 |
| 326.43 | 3.23 | 3.23 |
| 244.30 | 1.26 | 1.26 |
| 412.52 | 2.00 | 2.00 |
| 366.81 | 2.97 | 2.97 |
| 313.43 | 2.86 | 2.86 |
| 335.39 | 3.52 | 3.52 |