Basic Information
ID: ALA3720973
Type: Binding
Description: Inhibition of purified full-length human PASK expressed in insect cells using MBP protein substrate incubated for 10 mins before ATP addition and measured after 1 hr by kinase-Glo luminescent kinase assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA3720973
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 331.38 | 3.67 | 3.67 |
| 335.79 | 4.32 | 4.32 |
| 349.37 | 3.81 | 3.81 |
| 335.79 | 4.32 | 4.32 |
| 306.30 | 2.89 | 2.89 |
| 354.41 | 4.07 | 4.07 |
| 288.31 | 2.75 | 2.75 |
| 360.37 | 2.83 | 2.83 |
| 360.37 | 2.83 | 2.83 |
| 346.35 | 2.79 | 2.79 |
| 346.35 | 2.79 | 2.79 |
| 332.32 | 2.48 | 2.48 |
| 332.32 | 2.48 | 2.48 |
| 346.35 | 2.52 | 2.52 |
| 346.35 | 2.52 | 2.52 |
| 345.36 | 3.39 | 3.39 |
| 331.33 | 3.09 | 3.09 |
| 345.36 | 3.13 | 3.13 |
| 315.38 | 3.97 | 3.97 |
| 373.41 | 3.46 | 3.46 |
| 327.39 | 3.85 | 3.85 |
| 377.45 | 4.95 | 4.95 |
| 301.78 | 3.52 | 3.52 |
| 373.46 | 4.16 | 4.16 |
| 345.40 | 3.60 | 3.60 |
| 359.43 | 4.49 | 4.49 |
| 289.72 | 2.49 | 2.49 |
| 273.72 | 2.96 | 2.96 |
| 299.76 | 3.14 | 3.14 |
| 375.86 | 4.42 | 4.42 |
| 379.85 | 4.08 | 4.08 |
| 345.40 | 3.60 | 3.60 |
| 301.78 | 3.60 | 3.60 |
| 391.47 | 4.87 | 4.87 |
| 375.43 | 3.44 | 3.44 |
| 377.88 | 4.89 | 4.89 |
| 331.38 | 3.67 | 3.67 |
| 319.34 | 3.80 | 3.80 |
| 331.38 | 3.67 | 3.67 |
| 326.36 | 3.54 | 3.54 |
| 407.47 | 4.96 | 4.96 |
| 427.51 | 6.10 | 6.10 |
| 411.89 | 5.60 | 5.60 |
| 456.89 | 5.51 | 5.51 |
| 377.45 | 4.95 | 4.95 |
| 407.47 | 4.96 | 4.96 |
| 304.15 | 2.76 | 2.76 |
| 349.82 | 4.24 | 4.24 |
| 259.70 | 2.65 | 2.65 |
| 380.79 | 4.23 | 4.23 |