Assay Report Card

Basic Information

ID: ALA3721002

Type: Functional

Description: Antagonist activity against human P2X2/3 receptor expressed in CHOK1 cells assessed as inhibition of alpha,beta-meATP-induced calcium response incubated for 20 mins by Fluo-3AM dye based FLIPR assay

Organism: Homo sapiens

Cell type: CHO-K1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
400.223.173.17
444.272.992.99
458.303.383.38
458.303.383.38
458.303.383.38
474.302.352.35
474.302.352.35
488.332.602.60
472.333.773.77
298.352.552.55
458.303.383.38
284.322.242.24
342.402.372.37
356.432.762.76
356.432.762.76
372.431.731.73
356.432.762.76
353.401.211.21
427.480.400.40
478.723.003.00
404.643.813.81
488.332.742.74