Basic Information
ID: ALA3734107
Type: Binding
Description: Inhibition of GST/His6-tagged human YAK3 (124 to 526 residues) expressed in baculovirus infected insect Sf9 cells using biotinyl-LGGRDSRAGS*PMARR-OH as substrate after 2 hrs by scintillation proximity assay in presence of [gamma33P]ATP
Format: BAO_0000219
Organism: Homo sapiens
Cell type: Sf9
Target: Dual-specificity tyrosine-phosphorylation regulated kinase 3(ALA4575)
Document: ALA3733936
Inhibition of GST/His6-tagged human YAK3 (124 to 526 residues) expressed in baculovirus infected insect Sf9 cells using biotinyl-LGGRDSRAGS*PMARR-OH as substrate after 2 hrs by scintillation proximity assay in presence of [gamma33P]ATP: 38
Activity Charts
Bioactivity
Activity Types for Assay ALA3734107
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 410.30 | 4.89 | 4.89 |
| 380.86 | 4.55 | 4.55 |
| 365.85 | 4.78 | 4.78 |
| 390.39 | 4.53 | 4.53 |
| 326.43 | 2.36 | 2.36 |