Assay Report Card

Basic Information

ID: ALA3734121

Type: Binding

Description: Inhibition of full-length recombinant human GST-tagged ILK1 expressed in baculovirus infected insect Hi5 cells using CKRRRLASLR-amide as substrate after 15 mins by scintillation counting analysis in presence of [gamma-32P]-ATP

Organism: Homo sapiens

Cell type: BTI-TN-5B1-4

Activity Charts

Bioactivity

Activity Types for Assay ALA3734121

IC50

Total(152)

Compound Summary

Parent Molecular Weight	ALogP	Polar Surface Area
309.35	3.76	3.76
310.39	3.06	3.06
278.31	2.21	2.21
260.32	2.07	2.07
260.32	2.07	2.07
201.25	2.69	2.69
280.33	1.33	1.33
313.34	1.06	1.06
363.35	1.64	1.64
306.32	2.50	2.50
341.39	1.62	1.62
274.31	2.28	2.28
288.33	2.36	2.36
323.40	1.49	1.49
415.50	2.78	2.78
288.33	2.36	2.36
215.28	2.99	2.99
293.35	4.06	4.06
231.28	1.85	1.85
309.38	1.18	1.18
327.37	1.36	1.36
371.42	0.99	0.99
327.37	1.36	1.36
371.42	0.99	0.99
418.48	2.59	2.59
246.29	2.28	2.28
323.40	1.49	1.49
273.32	1.68	1.68
309.38	1.22	1.22
353.43	0.85	0.85
367.46	1.50	1.50
417.49	3.19	3.19
419.56	3.16	3.16
433.95	3.71	3.71
429.53	3.06	3.06
399.50	3.06	3.06
413.53	3.10	3.10
428.54	2.68	2.68
422.54	1.19	1.19
391.40	2.42	2.42
403.49	1.82	1.82
414.52	2.64	2.64
400.49	2.45	2.45
380.50	1.42	1.42
394.53	1.81	1.81
372.44	1.98	1.98
275.34	1.67	1.67
315.40	2.59	2.59
303.39	1.66	1.66
274.35	2.19	2.19
289.36	2.06	2.06
337.38	2.21	2.21
414.52	2.84	2.84
337.40	4.33	4.33
293.35	4.06	4.06
248.29	2.72	2.72
288.38	2.58	2.58
303.39	2.45	2.45
317.37	2.55	2.55
358.37	4.22	4.22
380.45	4.69	4.69
358.37	4.22	4.22
385.38	3.99	3.99
358.37	4.22	4.22
370.41	4.09	4.09
375.34	3.58	3.58
330.34	3.68	3.68
331.33	3.07	3.07
278.31	2.72	2.72
340.38	4.08	4.08
348.41	1.83	1.83
341.37	3.48	3.48
373.42	2.79	2.79
248.29	2.72	2.72
262.31	3.02	3.02
248.29	2.72	2.72
260.32	2.59	2.59
284.27	3.29	3.29
327.18	3.48	3.48
309.19	3.34	3.34
264.74	3.23	3.23
305.38	2.78	2.78
287.39	2.64	2.64
234.26	2.41	2.41
248.29	2.72	2.72
308.39	1.98	1.98
260.32	2.59	2.59
330.42	1.69	1.69
261.27	2.18	2.18
294.77	3.24	3.24
312.76	3.38	3.38
400.49	2.53	2.53
351.44	3.63	3.63
216.27	2.27	2.27
231.28	1.85	1.85
301.42	2.76	2.76
287.39	2.42	2.42
315.45	3.15	3.15
301.42	2.81	2.81
337.36	3.84	3.84
256.33	3.15	3.15
244.32	2.83	2.83
282.33	3.53	3.53
230.30	2.58	2.58
262.36	2.99	2.99
292.37	3.94	3.94
300.39	1.68	1.68
299.40	2.74	2.74
293.36	3.33	3.33
293.36	3.33	3.33
285.38	2.87	2.87
298.40	4.00	4.00
311.37	2.60	2.60
309.36	2.74	2.74
302.41	2.24	2.24
302.41	2.29	2.29
289.36	2.33	2.33
328.44	2.78	2.78
316.43	2.63	2.63
339.43	2.97	2.97
374.47	4.40	4.40
328.44	2.68	2.68
375.82	4.13	4.13
273.37	2.16	2.16
307.38	3.52	3.52
304.35	3.29	3.29
284.27	2.99	2.99
298.29	3.60	3.60
273.37	2.30	2.30
329.43	2.41	2.41
313.43	3.17	3.17
342.47	2.32	2.32
392.51	1.51	1.51
287.35	2.54	2.54
316.39	1.82	1.82
323.38	3.74	3.74
394.48	0.99	0.99
364.41	1.96	1.96
274.35	1.64	1.64
350.42	2.39	2.39
364.45	2.78	2.78
322.40	3.59	3.59
355.43	2.65	2.65
363.47	2.27	2.27
346.41	4.14	4.14
366.43	0.91	0.91
400.49	2.88	2.88
437.58	5.59	5.59
344.44	2.01	2.01
259.34	2.70	2.70
322.40	3.28	3.28
230.30	2.15	2.15