Inhibition of N-terminally GST-tagged human DLK catalytic domain (1 to 520 amino acids) using N- terminal His-tagged MKK4 K131M substrate incubated fo...

Basic Information

ID: ALA3734233

Type: Binding

Description: Inhibition of N-terminally GST-tagged human DLK catalytic domain (1 to 520 amino acids) using N- terminal His-tagged MKK4 K131M substrate incubated for 60 mins by TR-FRET assay

Format: BAO_0000357

Organism: Homo sapiens

Target: Mitogen-activated protein kinase kinase kinase 12(ALA1908389)

Document: ALA3727347

Inhibition of N-terminally GST-tagged human DLK catalytic domain (1 to 520 amino acids) using N- terminal His-tagged MKK4 K131M substrate incubated for 60 mins by TR-FRET assay: 38

Associated Items: Associated Bioactivities Associated Compounds

Activity Charts

Bioactivity

Activity Types for Assay ALA3734233

Total(503)

Compound Summary

Parent Molecular Weight	ALogP	Polar Surface Area
343.39	0.19	0.19
428.42	3.47	3.47
374.45	2.84	2.84
442.45	3.86	3.86
360.42	2.45	2.45
389.51	2.88	2.88
440.40	2.55	2.55
389.41	1.73	1.73
371.42	1.43	1.43
391.48	1.16	1.16
415.44	3.18	3.18
401.42	2.79	2.79
459.48	2.55	2.55
482.46	3.53	3.53
417.44	2.32	2.32
490.53	3.03	3.03
474.53	3.15	3.15
472.54	2.74	2.74
460.46	2.81	2.81
444.46	2.93	2.93
476.50	2.91	2.91
460.50	3.03	3.03
393.50	1.41	1.41
393.37	2.87	2.87
355.40	0.33	0.33
353.43	1.34	1.34
471.51	1.98	1.98
515.57	2.54	2.54
487.51	1.76	1.76
440.40	2.20	2.20
335.42	1.32	1.32
390.39	1.91	1.91
408.38	1.86	1.86
367.41	0.47	0.47
426.37	2.15	2.15
445.49	3.39	3.39
392.51	1.79	1.79
378.48	1.40	1.40
406.49	0.78	0.78
359.38	1.61	1.61
457.49	2.13	2.13
405.51	2.37	2.37
411.49	2.21	2.21
394.48	0.63	0.63
403.44	2.12	2.12
408.51	1.17	1.17
408.51	1.03	1.03
341.42	1.34	1.34
368.45	0.25	0.25
353.43	1.48	1.48
325.38	0.70	0.70
415.45	1.97	1.97
339.40	1.09	1.09
361.36	0.95	0.95
401.42	1.73	1.73
415.45	1.97	1.97
394.48	0.78	0.78
379.47	1.87	1.87
420.52	1.17	1.17
377.45	1.31	1.31
422.54	1.15	1.15
408.51	1.02	1.02
416.43	2.16	2.16
336.40	1.58	1.58
377.50	3.03	3.03
375.38	0.99	0.99
375.38	1.34	1.34
343.37	0.65	0.65
394.48	0.78	0.78
401.42	1.73	1.73
421.43	2.27	2.27
332.41	2.66	2.66
398.42	3.27	3.27
400.43	2.78	2.78
390.49	2.57	2.57
408.51	2.48	2.48
367.45	2.76	2.76
451.47	3.48	3.48
417.92	3.12	3.12
384.46	1.86	1.86
458.51	2.61	2.61
442.47	2.51	2.51
407.52	1.53	1.53
456.50	2.36	2.36
458.49	2.78	2.78
474.49	2.66	2.66
415.44	2.64	2.64
441.40	3.81	3.81
417.46	2.89	2.89
431.49	3.02	3.02
456.50	2.90	2.90
422.41	2.25	2.25
434.45	1.92	1.92
430.46	2.69	2.69
446.46	1.92	1.92
434.45	1.92	1.92
388.42	3.00	3.00
389.41	2.97	2.97
473.53	2.23	2.23
475.52	2.65	2.65