Basic Information
ID: ALA3734283
Type: Binding
Description: Inhibition of human GRK2 after 90 to 120 mins by Kinase-Glo assay
Format: BAO_0000357
Organism: Homo sapiens
Target: G-protein coupled receptor kinase 2(ALA4079)
Document: ALA3727367
Inhibition of human GRK2 after 90 to 120 mins by Kinase-Glo assay: 38
Activity Charts
Bioactivity
Activity Types for Assay ALA3734283
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 268.32 | 1.95 | 1.95 |
| 353.21 | 2.96 | 2.96 |
| 402.08 | 3.71 | 3.71 |
| 368.18 | 2.86 | 2.86 |
| 337.21 | 3.26 | 3.26 |
| 429.31 | 4.53 | 4.53 |
| 369.28 | 3.67 | 3.67 |
| 449.08 | 3.56 | 3.56 |
| 391.18 | 3.97 | 3.97 |
| 380.24 | 2.31 | 2.31 |
| 341.17 | 3.09 | 3.09 |
| 415.28 | 4.74 | 4.74 |
| 365.26 | 4.07 | 4.07 |
| 337.21 | 3.26 | 3.26 |
| 357.63 | 3.60 | 3.60 |
| 381.26 | 3.74 | 3.74 |
| 351.24 | 3.51 | 3.51 |
| 367.24 | 3.35 | 3.35 |
| 402.26 | 1.60 | 1.60 |
| 401.28 | 2.35 | 2.35 |
| 416.29 | 2.32 | 2.32 |
| 337.21 | 3.26 | 3.26 |
| 351.24 | 3.51 | 3.51 |
| 380.24 | 2.91 | 2.91 |
| 366.21 | 2.05 | 2.05 |
| 402.08 | 3.71 | 3.71 |
| 429.31 | 5.05 | 5.05 |
| 390.23 | 2.53 | 2.53 |
| 452.34 | 2.66 | 2.66 |
| 479.37 | 2.01 | 2.01 |
| 389.25 | 3.14 | 3.14 |
| 429.31 | 5.05 | 5.05 |
| 333.19 | 2.41 | 2.41 |
| 288.74 | 2.30 | 2.30 |
| 289.72 | 2.26 | 2.26 |
| 279.30 | 1.52 | 1.52 |
| 272.28 | 1.78 | 1.78 |
| 297.32 | 0.74 | 0.74 |
| 254.29 | 1.64 | 1.64 |
| 284.32 | 1.65 | 1.65 |
| 333.19 | 2.41 | 2.41 |
| 268.32 | 1.95 | 1.95 |
| 360.42 | 3.22 | 3.22 |
| 300.39 | 2.37 | 2.37 |
| 380.19 | 2.25 | 2.25 |
| 322.29 | 2.66 | 2.66 |
| 311.35 | 1.00 | 1.00 |
| 272.28 | 1.78 | 1.78 |
| 322.29 | 2.66 | 2.66 |
| 346.39 | 3.44 | 3.44 |
| 288.74 | 2.30 | 2.30 |
| 312.37 | 2.43 | 2.43 |
| 282.35 | 2.21 | 2.21 |
| 279.30 | 1.52 | 1.52 |
| 296.37 | 2.77 | 2.77 |
| 333.37 | 0.29 | 0.29 |
| 347.40 | 1.02 | 1.02 |
| 268.32 | 1.95 | 1.95 |
| 298.35 | 2.04 | 2.04 |
| 284.32 | 1.65 | 1.65 |
| 282.35 | 2.21 | 2.21 |
| 296.37 | 2.77 | 2.77 |
| 344.42 | 3.23 | 3.23 |
| 380.19 | 2.25 | 2.25 |
| 311.35 | 1.60 | 1.60 |
| 337.43 | 2.63 | 2.63 |
| 297.32 | 0.74 | 0.74 |
| 360.42 | 3.74 | 3.74 |
| 430.39 | 4.33 | 4.33 |
| 321.34 | 1.22 | 1.22 |
| 410.48 | 0.71 | 0.71 |
| 374.40 | 2.29 | 2.29 |
| 376.42 | 3.44 | 3.44 |
| 320.36 | 1.83 | 1.83 |
| 382.37 | 3.71 | 3.71 |
| 382.37 | 3.71 | 3.71 |
| 360.42 | 3.74 | 3.74 |
| 347.38 | 2.83 | 2.83 |
| 374.44 | 3.61 | 3.61 |
| 298.35 | 2.04 | 2.04 |
| 360.42 | 3.83 | 3.83 |
| 387.44 | 3.29 | 3.29 |
| 338.80 | 3.45 | 3.45 |
| 291.74 | 1.64 | 1.64 |
| 293.78 | 2.96 | 2.96 |
| 277.71 | 2.50 | 2.50 |
| 290.75 | 1.97 | 1.97 |
| 373.42 | 2.90 | 2.90 |
| 442.31 | 4.20 | 4.20 |
| 429.31 | 5.13 | 5.13 |
| 360.42 | 3.82 | 3.82 |
| 314.35 | 1.66 | 1.66 |
| 341.37 | 1.70 | 1.70 |
| 357.63 | 3.60 | 3.60 |
| 323.18 | 2.95 | 2.95 |
| 348.19 | 2.82 | 2.82 |
| 341.17 | 3.09 | 3.09 |