Basic Information
ID: ALA3736776
Type: Binding
Description: Inhibition of human recombinant haspin kinase domain expressed in Escherichia coli BL21-KRX using histone H3 (1 to 21) peptide substrate after 30 mins by scintillation and luminescence counting method in the presence of [gamma-33P]ATP
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA3736776
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 400.49 | 3.22 | 3.22 |
| 414.47 | 2.94 | 2.94 |
| 414.47 | 2.94 | 2.94 |
| 428.50 | 2.98 | 2.98 |
| 428.50 | 2.98 | 2.98 |
| 427.54 | 3.82 | 3.82 |
| 420.52 | 4.36 | 4.36 |
| 450.55 | 4.37 | 4.37 |
| 464.57 | 4.76 | 4.76 |
| 446.56 | 4.88 | 4.88 |
| 446.56 | 4.88 | 4.88 |
| 452.59 | 4.94 | 4.94 |
| 452.59 | 4.94 | 4.94 |
| 452.59 | 4.94 | 4.94 |
| 483.58 | 2.68 | 2.68 |
| 483.58 | 2.68 | 2.68 |
| 414.47 | 2.94 | 2.94 |
| 413.48 | 3.54 | 3.54 |
| 316.32 | 3.19 | 3.19 |
| 442.52 | 3.72 | 3.72 |
| 413.48 | 3.54 | 3.54 |