Basic Information
ID: ALA3737230
Type: Binding
Description: Inhibition of human recombinant LSD1/CoREST protein expressed in Escherichia coli using monomethylated H3-K4 peptide (21 amino acids) as substrate preincubated for 15 mins followed by substrate addition measured for 12 mins by HRP-coupled Ultrared detection system-based fluorescence analysis
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA3737230
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 465.98 | 3.98 | 3.98 |
| 415.92 | 3.24 | 3.24 |
| 375.86 | 2.37 | 2.37 |
| 277.75 | 2.08 | 2.08 |
| 395.89 | 3.44 | 3.44 |
| 410.91 | 3.19 | 3.19 |
| 424.93 | 2.87 | 2.87 |
| 411.89 | 3.74 | 3.74 |
| 411.89 | 3.74 | 3.74 |
| 327.82 | 3.23 | 3.23 |
| 445.95 | 4.59 | 4.59 |
| 460.97 | 4.35 | 4.35 |
| 474.99 | 4.02 | 4.02 |
| 461.95 | 4.89 | 4.89 |
| 461.95 | 4.89 | 4.89 |