Basic Information
ID: ALA3755178
Type: Binding
Description: Inhibition of mouse GAT1 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation counting
Organism: Mus musculus
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA3755178
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 127.14 | -0.01 | -0.01 |
| 505.61 | 4.82 | 4.82 |
| 350.42 | 3.17 | 3.17 |
| 153.22 | 1.60 | 1.60 |
| 139.24 | 2.07 | 2.07 |
| 167.21 | 0.78 | 0.78 |
| 288.14 | 1.41 | 1.41 |
| 193.29 | 2.50 | 2.50 |
| 207.27 | 2.02 | 2.02 |
| 249.27 | 0.76 | 0.76 |
| 221.26 | 1.20 | 1.20 |
| 274.16 | 2.23 | 2.23 |
| 229.71 | 2.08 | 2.08 |
| 278.40 | 2.32 | 2.32 |
| 292.42 | 2.71 | 2.71 |
| 294.40 | 1.56 | 1.56 |
| 364.49 | 2.50 | 2.50 |
| 280.41 | 2.57 | 2.57 |
| 293.41 | 1.13 | 1.13 |
| 321.16 | 2.27 | 2.27 |
| 236.28 | 2.15 | 2.15 |
| 260.17 | 2.71 | 2.71 |
| 264.41 | 2.80 | 2.80 |
| 278.44 | 3.19 | 3.19 |
| 280.41 | 2.03 | 2.03 |
| 350.50 | 2.98 | 2.98 |
| 334.46 | 2.51 | 2.51 |
| 266.43 | 3.04 | 3.04 |
| 279.43 | 1.61 | 1.61 |
| 336.39 | 0.30 | 0.30 |
| 335.40 | -0.13 | -0.13 |
| 406.48 | 1.24 | 1.24 |
| 197.23 | 0.56 | 0.56 |
| 237.30 | 1.46 | 1.46 |