Basic Information
ID: ALA3760353
Type: Binding
Description: Negative allosteric modulator activity at human CB1R expressed in CHO-K1 cells assessed as inhibition of CP55,940-induced beta-arrestin recruitment preincubated for 30 mins followed by CP55,940 addition measured for 90 mins by PathHunter assay relative to control
Organism: Homo sapiens
Cell type: CHO-K1
Activity Charts
Bioactivity
Activity Types for Assay ALA3760353
Emax
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 409.96 | 5.35 | 5.35 |
| 392.89 | 5.65 | 5.65 |
| 432.59 | 5.43 | 5.43 |
| 416.53 | 5.63 | 5.63 |
| 450.97 | 5.64 | 5.64 |
| 467.04 | 5.43 | 5.43 |
| 399.46 | 5.93 | 5.93 |
| 415.52 | 5.73 | 5.73 |
| 462.55 | 6.22 | 6.22 |