Assay Report Card

Basic Information

ID: ALA3760371

Type: Binding

Description: Positive allosteric modulator activity at human CB1R expressed in HEK293 cell membranes assessed as enhanced specific binding of [3H]CP55,940 at 500 nM pre-incubated for 60 mins before [3H]CP55,940 addition followed by drug wash-out by liquid scintillation spectrometric-based saturation binding assay

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
409.965.355.35
432.595.435.43