Antagonist activity at human TAAR1 receptor expressed in HEK293T cells cotransfected with beta-2 receptor assessed as inhibition of beta-PEA-induced c...

Basic Information

ID: ALA3772719

Type: Functional

Description: Antagonist activity at human TAAR1 receptor expressed in HEK293T cells cotransfected with beta-2 receptor assessed as inhibition of beta-PEA-induced cAMP production at 100 uM by BRET assay

Format: BAO_0000219

Organism: Homo sapiens

Cell type: HEK-293T

Target:  Trace amine-associated receptor 1(ALA5857)

Document:  ALA3769363

Antagonist activity at human TAAR1 receptor expressed in HEK293T cells cotransfected with beta-2 receptor assessed as inhibition of beta-PEA-induced cAMP production at 100 uM by BRET assay: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
226.282.552.55
232.241.491.49
202.261.211.21
192.220.510.51
347.253.923.92
308.433.513.51
333.233.183.18
334.403.833.83