ID: ALA3772988
Type: Binding
Description: Competitive inhibition of BRD4 in PMA /ionomycin activated human Jurkat cell lysate in presence of (S)-4-{3'-Cyano-4'-[3-(3-{2-[5-((3aR,6S,6aS)-2-oxo-hexahydro-thieno[3,4-d]imidazol-6-yl)-pentanoylamino]-ethyldisulfanyl}-propionylamino)-propoxy]-biphenyl-4-yl}-2,3,9-trimethyl-6H-1-thia-5,7,8,9a-tetraaza-cyclopenta[e]azulene-6-yl]acetic acid ethyl ester/avidin-resin by pull down assay
Format: BAO_0000219
Organism: Homo sapiens
Cell type: Jurkat
Target: Bromodomain-containing protein 4(ALA1163125)
Document: ALA3769406
Competitive inhibition of BRD4 in PMA /ionomycin activated human Jurkat cell lysate in presence of (S)-4-{3'-Cyano-4'-[3-(3-{2-[5-((3aR,6S,6aS)-2-oxo-hexahydro-thieno[3,4-d]imidazol-6-yl)-pentanoylamino]-ethyldisulfanyl}-propionylamino)-propoxy]-biphenyl-4-yl}-2,3,9-trimethyl-6H-1-thia-5,7,8,9a-tetraaza-cyclopenta[e]azulene-6-yl]acetic acid ethyl ester/avidin-resin by pull down assay: 1
Bioactivity
Activity Types for Assay ALA3772988
Inhibition
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
481.58 | 5.25 | 5.25 |
481.58 | 5.25 | 5.25 |