Basic Information
ID: ALA3776538
Type: Binding
Description: Inhibition of full length N-terminal His-tagged human recombinant LSD1 (1 to 852 residues) expressed in Escherichia coli BL21(DE3) cells using H3K4me2 peptide as substrate preincubated for 5 mins followed by substrate addition measured for 30 mins by peroxidase coupled assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA3776538
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 133.19 | 1.50 | 1.50 |
| 364.49 | 3.74 | 3.74 |
| 3762.38 | ||
| 2367.71 | ||
| 2404.77 | ||
| 3617.22 | ||
| 2480.87 | ||
| 3617.22 | ||
| 2482.88 | ||
| 2381.74 |