Basic Information
ID: ALA3776789
Type: Binding
Description: Inhibition of mouse GAT1 expressed in HEK293 cells assessed as remaining [3H]GABA uptake at 1 mM preincubated for 25 mins followed by [3H]GABA/unlabeled GABA addition measured after 4 mins by liquid scintillation counting analysis
Format: BAO_0000219
Organism: Mus musculus
Cell type: HEK293
Target: GABA transporter 1(ALA5445)
Document: ALA3774377
Inhibition of mouse GAT1 expressed in HEK293 cells assessed as remaining [3H]GABA uptake at 1 mM preincubated for 25 mins followed by [3H]GABA/unlabeled GABA addition measured after 4 mins by liquid scintillation counting analysis: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA3776789
Activity
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 185.27 | 1.49 | 1.49 |
| 183.25 | 1.26 | 1.26 |
| 181.24 | 0.71 | 0.71 |