Assay Report Card

Basic Information

ID: ALA3776791

Type: Binding

Description: Inhibition of mouse GAT4 expressed in HEK293 cells assessed as remaining [3H]GABA uptake at 1 mM preincubated for 25 mins followed by [3H]GABA/unlabeled GABA addition measured after 4 mins by liquid scintillation counting analysis

Organism: Mus musculus

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
185.271.491.49
183.251.261.26
181.240.710.71
195.261.101.10
211.302.042.04