Basic Information
ID: ALA3776820
Type: Binding
Description: Inhibition of human RORgamma ligand binding domain (Serine 253 to Lysine 518 residues) expressed in CHOK1 cells incubated for 2 days by Gal4 luciferase reporter gene assay
Organism: Homo sapiens
Cell type: CHO-K1
Activity Charts
Bioactivity
Activity Types for Assay ALA3776820
EC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 428.56 | 5.06 | 5.06 |
| 412.49 | 4.35 | 4.35 |
| 410.52 | 4.90 | 4.90 |
| 424.55 | 5.47 | 5.47 |
| 424.55 | 5.15 | 5.15 |
| 426.52 | 4.40 | 4.40 |
| 376.50 | 5.07 | 5.07 |
| 390.53 | 5.15 | 5.15 |
| 404.56 | 5.54 | 5.54 |
| 364.49 | 4.61 | 4.61 |
| 378.52 | 5.00 | 5.00 |
| 398.51 | 4.81 | 4.81 |
| 402.97 | 5.34 | 5.34 |
| 382.55 | 5.00 | 5.00 |
| 382.55 | 5.00 | 5.00 |
| 394.56 | 5.31 | 5.31 |
| 408.59 | 5.70 | 5.70 |
| 430.54 | 5.56 | 5.56 |
| 368.53 | 4.78 | 4.78 |
| 368.53 | 4.78 | 4.78 |
| 382.55 | 5.17 | 5.17 |
| 416.57 | 5.67 | 5.67 |
| 407.52 | 4.65 | 4.65 |
| 394.56 | 5.34 | 5.34 |
| 394.56 | 5.34 | 5.34 |
| 463.67 | 5.44 | 5.44 |
| 450.63 | 5.26 | 5.26 |
| 477.65 | 4.97 | 4.97 |