ID: ALA3778806
Type: Binding
Description: Inhibition of recombinant human N-terminal GST-tagged KDM4B (1 to 500 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 as substrate preincubated for 10 mins measured after 20 mins by alphascreen assay
Organism: Homo sapiens
Cell type: Sf9
Bioactivity
Activity Types for Assay ALA3778806
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
281.34 | 3.46 | 3.46 |
359.43 | 2.86 | 2.86 |
373.46 | 3.25 | 3.25 |
373.46 | 3.25 | 3.25 |
147.14 | 0.32 | 0.32 |
221.24 | 1.49 | 1.49 |
220.26 | 0.89 | 0.89 |
206.23 | 1.90 | 1.90 |
220.25 | 2.21 | 2.21 |
325.35 | 3.16 | 3.16 |
238.17 | 1.66 | 1.66 |
248.21 | 2.07 | 2.07 |
245.27 | 1.02 | 1.02 |
230.25 | 1.44 | 1.44 |
213.20 | 0.71 | 0.71 |
227.23 | 0.72 | 0.72 |
213.20 | 0.50 | 0.50 |
266.30 | 1.61 | 1.61 |
256.26 | 1.20 | 1.20 |
259.31 | 0.07 | 0.07 |
204.23 | 0.38 | 0.38 |
244.30 | 1.30 | 1.30 |
321.38 | 1.64 | 1.64 |
322.37 | 1.04 | 1.04 |
257.25 | 0.04 | 0.04 |
284.32 | 0.61 | 0.61 |
310.36 | 1.14 | 1.14 |
324.39 | 1.53 | 1.53 |
378.41 | 2.32 | 2.32 |
429.31 | 3.49 | 3.49 |
438.51 | 1.58 | 1.58 |
385.43 | 2.05 | 2.05 |
399.46 | 2.44 | 2.44 |
448.96 | 3.65 | 3.65 |
414.51 | 3.00 | 3.00 |
432.50 | 3.14 | 3.14 |
482.51 | 4.02 | 4.02 |
483.40 | 4.31 | 4.31 |
444.54 | 3.01 | 3.01 |
458.52 | 2.73 | 2.73 |
415.50 | 2.40 | 2.40 |
446.52 | 2.26 | 2.26 |
434.93 | 3.58 | 3.58 |
418.48 | 3.07 | 3.07 |
430.51 | 2.93 | 2.93 |
478.58 | 2.33 | 2.33 |
425.50 | 2.80 | 2.80 |
434.93 | 3.58 | 3.58 |
400.49 | 2.93 | 2.93 |
401.47 | 2.32 | 2.32 |
406.52 | 2.99 | 2.99 |
469.38 | 4.23 | 4.23 |
434.93 | 3.58 | 3.58 |
436.47 | 3.20 | 3.20 |
436.47 | 3.20 | 3.20 |
468.48 | 3.94 | 3.94 |