Assay Report Card

Basic Information

ID: ALA3778806

Type: Binding

Description: Inhibition of recombinant human N-terminal GST-tagged KDM4B (1 to 500 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 as substrate preincubated for 10 mins measured after 20 mins by alphascreen assay

Organism: Homo sapiens

Cell type: Sf9

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
281.343.463.46
359.432.862.86
373.463.253.25
373.463.253.25
147.140.320.32
221.241.491.49
220.260.890.89
206.231.901.90
220.252.212.21
325.353.163.16
238.171.661.66
248.212.072.07
245.271.021.02
230.251.441.44
213.200.710.71
227.230.720.72
213.200.500.50
266.301.611.61
256.261.201.20
259.310.070.07
204.230.380.38
244.301.301.30
321.381.641.64
322.371.041.04
257.250.040.04
284.320.610.61
310.361.141.14
324.391.531.53
378.412.322.32
429.313.493.49
438.511.581.58
385.432.052.05
399.462.442.44
448.963.653.65
414.513.003.00
432.503.143.14
482.514.024.02
483.404.314.31
444.543.013.01
458.522.732.73
415.502.402.40
446.522.262.26
434.933.583.58
418.483.073.07
430.512.932.93
478.582.332.33
425.502.802.80
434.933.583.58
400.492.932.93
401.472.322.32
406.522.992.99
469.384.234.23
434.933.583.58
436.473.203.20
436.473.203.20
468.483.943.94