Basic Information
ID: ALA3779310
Type: Binding
Description: Inhibition of recombinant human His-tagged TRIM24-PHD/bromodomain expressed in Escherichia coli strains BL21 (DE3) cells using biotinylated H3K23ac (1 to 33 residues) peptide after 1 hr by AlphaScreen assay
Organism: Homo sapiens
Cell type: BL21-DE3
Activity Charts
Bioactivity
Activity Types for Assay ALA3779310
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 372.41 | 1.56 | 1.56 |
| 347.40 | 1.69 | 1.69 |
| 317.37 | 1.68 | 1.68 |
| 439.49 | 3.48 | 3.48 |
| 244.32 | 2.64 | 2.64 |
| 348.45 | 2.73 | 2.73 |
| 362.48 | 3.12 | 3.12 |
| 362.48 | 3.12 | 3.12 |
| 376.43 | 2.41 | 2.41 |
| 388.49 | 3.43 | 3.43 |
| 398.53 | 4.44 | 4.44 |
| 346.41 | 2.40 | 2.40 |
| 363.46 | 2.40 | 2.40 |
| 389.48 | 2.71 | 2.71 |
| 399.52 | 3.73 | 3.73 |
| 519.58 | 3.78 | 3.78 |
| 519.58 | 3.78 | 3.78 |
| 575.64 | 5.07 | 5.07 |
| 533.61 | 4.09 | 4.09 |
| 471.54 | 2.91 | 2.91 |
| 527.60 | 4.28 | 4.28 |
| 485.57 | 3.30 | 3.30 |
| 499.59 | 3.55 | 3.55 |
| 499.59 | 3.69 | 3.69 |
| 445.54 | 3.61 | 3.61 |
| 326.40 | 3.70 | 3.70 |
| 515.59 | 2.93 | 2.93 |
| 513.58 | 2.62 | 2.62 |
| 584.70 | 4.21 | 4.21 |
| 686.83 | 5.46 | 5.46 |
| 586.72 | 3.89 | 3.89 |
| 587.70 | 3.92 | 3.92 |
| 642.78 | 5.17 | 5.17 |
| 572.69 | 3.50 | 3.50 |
| 558.66 | 3.11 | 3.11 |
| 614.72 | 4.39 | 4.39 |
| 600.69 | 4.00 | 4.00 |
| 642.78 | 5.00 | 5.00 |