Assay Report Card

Basic Information

ID: ALA3782666

Type: Binding

Description: Binding affinity to human His6-tagged BRDT bromodomain 1 (N21 to E137 residues) expressed in Escherichia coli BL21(DE3) cells at 200 uM incubated for 30 mins by SYPRO orange staining based fluorescence thermal shift assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
457.005.535.53
404.452.352.35
415.522.362.36
509.055.485.48
396.423.323.32
370.413.763.76
318.402.512.51
447.563.403.40
358.463.433.43
416.551.741.74
332.433.363.36
358.463.893.89
370.403.763.76
388.393.903.90
416.894.284.28
461.344.394.39