Inhibition of human GLUT3 expressed in GLUT1 knock-out DLD1 cells assessed as ATP production co-incubated with 300 mM glucose for 16 hrs by CellTiter-...

Basic Information

ID: ALA3782732

Type: Binding

Description: Inhibition of human GLUT3 expressed in GLUT1 knock-out DLD1 cells assessed as ATP production co-incubated with 300 mM glucose for 16 hrs by CellTiter-Glo assay in presence of oxidative phosphorylation inhibitor rotenone

Format: BAO_0000219

Organism: Homo sapiens

Cell type: DLD-1

Target: Solute carrier family 2, facilitated glucose transporter member 3(ALA5215)

Document: ALA3779893

Inhibition of human GLUT3 expressed in GLUT1 knock-out DLD1 cells assessed as ATP production co-incubated with 300 mM glucose for 16 hrs by CellTiter-Glo assay in presence of oxidative phosphorylation inhibitor rotenone: 1

Associated Items: Associated Bioactivities Associated Compounds

Activity Charts

Bioactivity

Activity Types for Assay ALA3782732

IC50

Total(57)

Compound Summary

Parent Molecular Weight	ALogP	Polar Surface Area
400.49	3.46	3.46
374.42	3.28	3.28
372.43	2.85	2.85
386.46	3.15	3.15
440.43	4.04	4.04
381.44	3.01	3.01
424.43	4.16	4.16
374.42	3.28	3.28
386.46	3.15	3.15
381.44	3.01	3.01
386.46	3.15	3.15
404.45	3.29	3.29
411.47	3.02	3.02
404.45	3.29	3.29
411.47	3.02	3.02
404.45	3.29	3.29
411.47	3.02	3.02
429.48	2.25	2.25
404.45	3.29	3.29
387.45	2.55	2.55
387.45	2.55	2.55
387.45	2.55	2.55
387.45	2.55	2.55
378.48	2.24	2.24
385.47	4.21	4.21
385.47	4.21	4.21
400.49	3.54	3.54
400.49	3.54	3.54
398.47	3.29	3.29
398.47	3.29	3.29
398.47	3.15	3.15
400.49	3.54	3.54
385.47	3.76	3.76
385.47	3.76	3.76
387.45	2.55	2.55
387.45	2.55	2.55
386.46	3.15	3.15
402.46	2.44	2.44
404.45	3.29	3.29
416.49	3.16	3.16
400.49	3.46	3.46
404.45	3.29	3.29
411.47	3.02	3.02
416.49	3.16	3.16
400.49	3.46	3.46
404.45	3.29	3.29
411.47	3.02	3.02
416.49	3.16	3.16
422.44	3.43	3.43
434.48	3.30	3.30
414.51	3.77	3.77
387.45	2.55	2.55
387.45	2.55	2.55
387.45	2.55	2.55
405.44	2.68	2.68
417.47	2.55	2.55
378.48	3.28	3.28