Assay Report Card

Basic Information

ID: ALA3782932

Type: Binding

Description: Inhibition of N-terminal GST-tagged recombinant human FGFR1 (456 to 765 residues) expressed in baculovirus infected insect Sf21 cells after 25 mins using KKKSPGEYVNIEFG peptide substrate by scintillation counting analysis

Organism: Homo sapiens

Cell type: Sf21

Activity Charts

Bioactivity

Activity Types for Assay ALA3782932

IC50

Total(25)

Compound Summary

Parent Molecular Weight	ALogP	Polar Surface Area
308.32	2.42	2.42
290.33	2.28	2.28
320.35	2.29	2.29
304.35	2.59	2.59
304.35	2.59	2.59
320.35	2.29	2.29
320.35	2.29	2.29
334.38	2.68	2.68
350.38	2.30	2.30
350.38	2.30	2.30
348.41	2.90	2.90
354.80	2.94	2.94
324.77	2.93	2.93
338.80	3.24	3.24
322.34	2.73	2.73
324.77	2.93	2.93
308.32	2.42	2.42
338.80	3.24	3.24
358.32	3.30	3.30
306.33	1.99	1.99
320.35	2.00	2.00
320.35	2.29	2.29
320.35	2.00	2.00
320.35	2.29	2.29
306.33	1.99	1.99