Basic Information
ID: ALA3787887
Type: Binding
Description: Inhibition of GST fused human recombinant DYRK1A expressed in Escherichia coli using woodtide as substrate after 30 mins by scintillation counting in presence of [gamma33P]ATP
Format: BAO_0000019
Organism: Homo sapiens
Target: Dual-specificity tyrosine-phosphorylation regulated kinase 1A(ALA2292)
Document: ALA3784980
Inhibition of GST fused human recombinant DYRK1A expressed in Escherichia coli using woodtide as substrate after 30 mins by scintillation counting in presence of [gamma33P]ATP: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA3787887
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 322.37 | 3.41 | 3.41 |
| 323.36 | 2.80 | 2.80 |
| 336.40 | 3.71 | 3.71 |
| 380.40 | 3.19 | 3.19 |
| 336.40 | 3.71 | 3.71 |
| 352.39 | 2.90 | 2.90 |
| 366.42 | 3.55 | 3.55 |
| 421.50 | 3.24 | 3.24 |
| 434.54 | 3.15 | 3.15 |
| 419.53 | 4.39 | 4.39 |
| 336.40 | 3.71 | 3.71 |
| 336.40 | 3.71 | 3.71 |
| 350.38 | 3.22 | 3.22 |
| 380.40 | 3.19 | 3.19 |
| 352.39 | 2.90 | 2.90 |
| 366.42 | 3.55 | 3.55 |
| 421.50 | 3.24 | 3.24 |
| 434.54 | 3.15 | 3.15 |
| 419.53 | 4.39 | 4.39 |
| 405.50 | 4.00 | 4.00 |
| 407.52 | 4.25 | 4.25 |
| 337.38 | 3.11 | 3.11 |
| 337.38 | 3.11 | 3.11 |
| 337.38 | 3.11 | 3.11 |
| 372.43 | 4.56 | 4.56 |
| 402.45 | 4.57 | 4.57 |
| 354.39 | 3.88 | 3.88 |