Basic Information
ID: ALA3788932
Type: Binding
Description: Inhibition of recombinant human C-terminal FLAG-tagged KDM5A (1 to 1090 residues) expressed in baculovirus infected sf9 cells using biotin-H3K4me3 substrate incubated for 30 mins by TR-FRET assay
Organism: Homo sapiens
Cell type: Sf9
Activity Charts
Bioactivity
Activity Types for Assay ALA3788932
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 203.20 | 1.18 | 1.18 |
| 309.33 | 2.86 | 2.86 |
| 349.39 | 3.64 | 3.64 |
| 227.23 | 0.66 | 0.66 |
| 329.74 | 3.20 | 3.20 |
| 343.77 | 3.51 | 3.51 |
| 357.34 | 2.22 | 2.22 |
| 286.38 | 3.41 | 3.41 |
| 340.36 | 4.13 | 4.13 |
| 269.26 | 1.81 | 1.81 |
| 352.37 | 3.18 | 3.18 |
| 332.74 | 3.50 | 3.50 |
| 372.81 | 4.28 | 4.28 |
| 386.71 | 4.39 | 4.39 |