Basic Information
ID: ALA3788935
Type: Binding
Description: Inhibition of recombinant human N-terminal His-tagged KDM4A (1 to 350 residues) expressed in Escherichia coli using biotin-H3K9me3 substrate incubated for 30 mins by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA3788935
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 203.20 | 1.18 | 1.18 |
| 227.23 | 0.66 | 0.66 |
| 332.74 | 3.50 | 3.50 |
| 372.81 | 4.28 | 4.28 |
| 386.71 | 4.39 | 4.39 |