Assay Report Card

Basic Information

ID: ALA3794937

Type: Binding

Description: Inhibition of full length human N-terminal GST-tagged MAPKAPK2 (1 to 400 residues) expressed in baculovirus expression system coexpressing human His-tagged p38beta (1 to 364 residues)/MAP2K6 (1 to 334 residues) using fluorescence labelled GS peptide substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
237.262.822.82
425.493.783.78
411.514.144.14