Assay Report Card

Basic Information

ID: ALA3794940

Type: Binding

Description: Inhibition of full length human N-terminal His-tagged NEK2 (1 to 445 residues) expressed in baculovirus expression system using fluorescence labelled CDK7 peptide substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
237.262.822.82
425.493.783.78
411.514.144.14