Assay Report Card

Basic Information

ID: ALA3794950

Type: Binding

Description: Inhibition of human N-terminal GST-tagged ROCK1 catalytic domain (1 to 477 residues) expressed in baculovirus expression system using fluorescence labelled LIMKtide substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
237.262.822.82
425.493.783.78
411.514.144.14