Assay Report Card

Basic Information

ID: ALA3795199

Type: Binding

Description: Binding affinity to FKBP51 FK506-binding domain (1 to 140 amino acids) (unknown origin) incubated for 30 mins using fluorescein-conjugated 2-(5-((2-(3-((R)-3-(3,4-dimethoxyphenyl)-1-((S)-1-(3,3-dimethyl-2-oxopentanoyl)piperidine-2-carbonyloxy)propyl)phenoxy)acetamido)methyl)-6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic acid by competitive fluorescence polarization assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
746.906.736.73
446.593.893.89
475.592.362.36
489.612.752.75
503.643.143.14
517.673.533.53
489.612.752.75
489.612.752.75
503.643.143.14
503.643.143.14
503.643.143.14
517.673.533.53
517.673.383.38
517.673.383.38
531.693.773.77
531.693.773.77
531.693.773.77
557.734.314.31
551.684.104.10
551.684.104.10
565.713.973.97
565.713.973.97
571.764.704.70
579.744.364.36
585.795.095.09
505.611.721.72
505.611.721.72
519.642.112.11
519.642.112.11
546.671.991.99
546.671.991.99
555.682.692.69
555.682.692.69
501.622.892.89
515.653.283.28
529.683.673.67
543.714.064.06
545.682.912.91
586.732.792.79